Amoxapine — Mechanism Gap Analysis
HYPOTHESIS_ENGINE_v1.0 · Corpus v20260227-01 · Deterministic graph-traversal
Known Targets
CYP2C19CYP2D6ARCYP2C9ESR1CYTOCHROMETDP1CYP1A2THRBCYP3A4CYP3A7SYKTYROSINE-PROTEINGLI3PGRTP53NR3C1ABCB1KCNH2CHRM1DRD35-HYDROXYTRYPTAMINEADRA1AHTR2ADRD2DRD1CYP19A1HTR1AADRA2AADRB2VDRHTR2BADRA2CJUNADRA2BATXN2SLC6A3PMP22SLC6A4MU-TYPESLC6A2HTR2CKAPPA-TYPESODIUM-DEPENDENTCHRM2HRH1ALPHA-2ACHRM5CHRM3ALPHA-2BHRH2HTR7HTR6ALPHA-1DHTTALPHA-1AALPHA-2CDRD4ALPHA-1BKCNMB1KCNMB2MUSCARINICHTR5AHISTAMINEPDE4DTHPOKCNMA1DRD5HTR3ATRPC6TRPC4TACR1DELTA-TYPENPR2HRH4
75 known targets mapped from PubChem bioassay data
Pathway Context
Class A/1 (Rhodopsin-like receptors)24 targets overlapping
Amine ligand-binding receptors23 targets overlapping
Hemostasis10 targets overlapping
Uncovered Pathway Targets
299 totalADORA2BADORA3ADRA1BADRA1DADRB1ADRB3AGTR1AGTR2APLNRAPP+289 more…
Genes present in the top pathway union that Amoxapine does not directly modulate.
Top Stack Candidates
Isoproterenol Isopropyl analog of EPINEPHRINE; beta-sympathomimetic that acts on
score 9,410.826#1 gap-filler · 31 targets covered · evidence score 44.3
ADRA1BADRA1DADRB1ADRB3TSHRCREB1GRK2TAS2R1TAS2R10TAS2R13TAS2R14TAS2R16+19
Sorafenib
score 5,251.01#2 gap-filler · 21 targets covered · evidence score 44.4
ADORA3MLNRABL1CDK5CSKFGRFYNIFNB1LCKLYNMAPK1MAPK14+9
679 more candidates · full stack optimisation locked
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BiohacksAI maps biological mechanisms. It does not recommend compounds. Results generated by HYPOTHESIS_ENGINE_v1.0.