Cyproheptadine — Mechanism Gap Analysis
HYPOTHESIS_ENGINE_v1.0 · Corpus v20260227-01 · Deterministic graph-traversal
Known Targets
CYP2C19CYP2D6ARTDP1THRBCYP3A7SYKTYROSINE-PROTEINGLI3RATTUSNSD2MUSHISTONE-LYSINEKCNH2RARACHRM1DRD35-HYDROXYTRYPTAMINEADRA1AHTR2ADRD2DRD1HTR1AADRA2AHTR2BJUNSLC6A4SLC6A2HTR2CSODIUM-DEPENDENTCHRM2HRH1ALPHA-2ACHRM5CHRM4ADRA1BADRA1DCHRM3ALPHA-2BHTR7HTR6ALPHA-1DALPHA-1AALPHA-2CDRD4ALPHA-1BHTR1BMUSCARINICHTR1DSCN2AHTR5AHISTAMINESCN3ASCN1AHTR1FDRD5HTR3ANPR2HTR3BHTR4EHMT2HTR5BSETD7SUV39H1DOT1LKMT5A
66 known targets mapped from PubChem bioassay data
Pathway Context
Class A/1 (Rhodopsin-like receptors)22 targets overlapping
Amine ligand-binding receptors22 targets overlapping
G alpha (q) signalling events10 targets overlapping
Uncovered Pathway Targets
193 totalADORA2BADORA3ADRA2BADRA2CADRB1ADRB2ADRB3AGTR1AGTR2APLNR+183 more…
Genes present in the top pathway union that Cyproheptadine does not directly modulate.
Top Stack Candidates
s adenosylhomocysteine
score 5,279.182#1 gap-filler · 17 targets covered · evidence score 43.5
ASH2LCARM1DPY30EHMT1EZH2KMT2AKMT5CPRMT1PRMT3PRMT5PRMT6PRMT7+5
Astemizole Antihistamine drug now withdrawn from
score 4,340.789#2 gap-filler · 17 targets covered · evidence score 48.7
ADRA2CADRB2APLNRAVPR1AGALR2GHSRHRH2HRH4MLNROXTRSSTR5TAAR1+5
611 more candidates · full stack optimisation locked
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BiohacksAI maps biological mechanisms. It does not recommend compounds. Results generated by HYPOTHESIS_ENGINE_v1.0.