Amlodipine — Mechanism Gap Analysis
HYPOTHESIS_ENGINE_v1.0 · Corpus v20260227-01 · Deterministic graph-traversal
Known Targets
CYP2D6CYP2C9CYP3A7CHRM1DRD3ADRA1ADRD2ADRA2AADRB2HTR2BADRA2CSLC6A3SLC6A2ADRA1BADRA1DHRH2HTR6TBXA2RCACNA1CHTR3ACACNA1DKCNK2NAE1UBE2M
24 known targets mapped from PubChem bioassay data
Pathway Context
Class A/1 (Rhodopsin-like receptors)13 targets overlapping
Amine ligand-binding receptors12 targets overlapping
G alpha (q) signalling events6 targets overlapping
Uncovered Pathway Targets
177 totalADORA2BADORA3ADRA2BADRB1ADRB3AGTR1AGTR2APLNRAPPAVPR1A+167 more…
Genes present in the top pathway union that Amlodipine does not directly modulate.
Top Stack Candidates
Astemizole Antihistamine drug now withdrawn from
score 4,787.062#1 gap-filler · 21 targets covered · evidence score 48.7
APLNRAVPR1ACHRM2CHRM3DRD1DRD4GALR2GHSRHRH1HRH4HTR1AHTR2A+9
Aripiprazole
score 4,678.224#2 gap-filler · 21 targets covered · evidence score 52.0
ADORA3ADRA2BADRB1ADRB3AGTR1AVPR1ACHRM2DRD1DRD4DRD5HRH1HRH3+9
668 more candidates · full stack optimisation locked
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BiohacksAI maps biological mechanisms. It does not recommend compounds. Results generated by HYPOTHESIS_ENGINE_v1.0.