Carvedilol — Mechanism Gap Analysis
HYPOTHESIS_ENGINE_v1.0 · Corpus v20260227-01 · Deterministic graph-traversal
Known Targets
NR1I2CHAINRATTUSRORCABCB1KCNH2DRD35-HYDROXYTRYPTAMINEADRA1ADRD2DRD1HTR1AADRA2AADRB2HTR2BADRA2CADRA2BSLC6A3SLC6A4MU-TYPESLC6A2HTR2CSODIUM-DEPENDENTALPHA-2AADRB1ADRA1BADRA1DALPHA-2BHRH2HTR7HTR6ALPHA-1DALPHA-1AALPHA-2CDRD4BAZ2BALPHA-1BKCNMB1KCNMB2ADRB3PTGER2MAP4K2KCNMB4NPY1RKCNMA1GRIN1CYP1B1SCN5ASLC22A1SLC22A2BETA-1KCNJ2NPY2RTRPC6HCRTR1TRPC4TACR1BETA-3BETA-2AGTR1LRRC26OXTRMLNRVOLTAGE-GATEDKCNK2KCNK10
66 known targets mapped from PubChem bioassay data
Pathway Context
Class A/1 (Rhodopsin-like receptors)27 targets overlapping
Amine ligand-binding receptors19 targets overlapping
Neuronal System11 targets overlapping
Uncovered Pathway Targets
262 totalADORA2BADORA3AGTR2APLNRAPPAVPR1AAVPR1BAVPR2BDKRB1BDKRB2+252 more…
Genes present in the top pathway union that Carvedilol does not directly modulate.
Top Stack Candidates
Ondansetron
score 6,579.264#1 gap-filler · 23 targets covered · evidence score 56.7
CCKBRCHRM1HTR2AHTR4OPRM1ACHECHRNA4GABRA1GABRA2GABRA3GABRA4GABRA5+11
Colchicine
score 5,037.002#2 gap-filler · 21 targets covered · evidence score 42.1
CXCL8GLRA1GLRA2MDM2TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBA8TUBAL3+9
700 more candidates · full stack optimisation locked
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BiohacksAI maps biological mechanisms. It does not recommend compounds. Results generated by HYPOTHESIS_ENGINE_v1.0.