Fluspirilene — Mechanism Gap Analysis
HYPOTHESIS_ENGINE_v1.0 · Corpus v20260227-01 · Deterministic graph-traversal
Known Targets
CYP2D6ARCYP2C9ESR1TDP1CYP1A2THRBESRRACHAINPGRNSD2RORCHISTONE-LYSINENUCLEARKCNH2RARAEUCHROMATICDRD35-HYDROXYTRYPTAMINEADRA1AHTR2ADRD2ESR2HTR1AIFNGPPARGADRB2HTR2BADRA2CADRA2BATXN2ATAD5SLC6A3PMP22SLC6A4MU-TYPESLC6A2SMAD3KAPPA-TYPEGMNNSTK33HRH1MDM2MDM4OPRM1IFNB1IDH1ADORA3CHRM3HTR6PPARDOPRD1HTTBRCA1HTR1DPPP1R15AGPR151CBX1BARD1CACNA1CTHPOMPHOSPH8MAP4K2HTR1ETAAR1NPSR1APAF1TRPC6HCRTR1TRPC4DELTA-TYPEGHSRPPP1CADDIT3ABHD4MLNRMC3RGLRA1GNA15KCNK2MAP1LC3AXBP1NTSR1OPRL1
84 known targets mapped from PubChem bioassay data
Pathway Context
Class A/1 (Rhodopsin-like receptors)24 targets overlapping
Amine ligand-binding receptors14 targets overlapping
G alpha (q) signalling events12 targets overlapping
Uncovered Pathway Targets
200 totalADORA2BADRA1BADRA1DADRA2AADRB1ADRB3AGTR1AGTR2APLNRAPP+190 more…
Genes present in the top pathway union that Fluspirilene does not directly modulate.
Top Stack Candidates
Isoproterenol Isopropyl analog of EPINEPHRINE; beta-sympathomimetic that acts on
score 9,597.5#1 gap-filler · 32 targets covered · evidence score 44.3
ADRA1BADRA1DADRB1ADRB3DRD4TSHRCREB1GRK2TAS2R1TAS2R10TAS2R13TAS2R14+20
Aripiprazole
score 4,138.317#2 gap-filler · 19 targets covered · evidence score 52.0
ADRA1BADRA1DADRA2AADRB1ADRB3AGTR1AVPR1ACHRM1CHRM2DRD1DRD4DRD5+7
645 more candidates · full stack optimisation locked
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BiohacksAI maps biological mechanisms. It does not recommend compounds. Results generated by HYPOTHESIS_ENGINE_v1.0.