EIF2AK2
MOLECULAR TARGETeukaryotic translation initiation factor 2 alpha kinase 2
EIF2AK2 (eukaryotic translation initiation factor 2 alpha kinase 2) is targeted by 25 compounds in the BiohacksAI evidence corpus, derived from PubMed bioassay data. Each compound is ranked by confidence score (log-normalized assay count × evidence quality).
Compounds Targeting EIF2AK2
Ranked by bioassay confidence score (PubChem active assay count × evidence quality).
| # | Compound | Confidence | Active Assays |
|---|---|---|---|
| 1 | erlotinib | 5.55 | 256 |
| 2 | alvocidib | 4.52 | 91 |
| 3 | bi 2536 | 4.01 | 54 |
| 4 | midostaurin | 3.85 | 46 |
| 5 | pazopanib | 3.69 | 39 |
| 6 | pelitinib | 3.50 | 32 |
| 7 | 6bio | 3.50 | 32 |
| 8 | fedratinib | 3.40 | 29 |
| 9 | sp 600125 | 3.22 | 24 |
| 10 | dorsomorphin | 3.14 | 22 |
| 11 | dovitinib | 3.09 | 21 |
| 12 | jnj 7706621 | 3.09 | 21 |
| 13 | lestaurtinib | 3.04 | 20 |
| 14 | r 406 | 2.83 | 16 |
| 15 | su 9516 | 2.83 | 16 |
| 16 | kw 2449 | 2.64 | 13 |
| 17 | gsk 690693 | 2.64 | 13 |
| 18 | ast 487 | 2.56 | 12 |
| 19 | raf 265 | 2.48 | 11 |
| 20 | su 014813 | 2.20 | 8 |
| 21 | anilinopyrimidine1 | 1.79 | 5 |
| 22 | quinoxaline1 | 1.79 | 5 |
| 23 | Axitinib | 0.69 | 1 |
| 24 | Crizotinib | 0.69 | 1 |
| 25 | sp600125 | 0.69 | 1 |
About EIF2AK2 as a Drug Target
EIF2AK2 (eukaryotic translation initiation factor 2 alpha kinase 2) is a well-characterized molecular target in biomedical research. BiohacksAI tracks 25 compounds with documented EIF2AK2 interaction from PubChem bioassay data, cross-referenced with PubMed clinical evidence. The confidence score reflects the log-normalized count of active PubChem assays, weighted by evidence quality from the BiohacksAI corpus.
EIF2AK2 inhibitors, activators, and modulators are of interest in research areas including longevity, metabolic health, and neurological function. Each compound profile includes evidence score, RCT count, human study ratio, research velocity, and domain relevance.