Molecular Targets
Browse 500 molecular targets with compound interaction data from PubChem bioassays. Each target page lists all compounds that interact with the target, ranked by bioassay confidence score.
Most-Targeted Genes
CYP2C19334 compoundsCYP2D6324 compoundsAR296 compoundsCYP2C9295 compoundsNR1I2259 compoundsESR1253 compoundsCYTOCHROME244 compoundsTDP1241 compoundsCYP1A2230 compoundsTHRB230 compoundsESRRA227 compoundsCYP3A4224 compoundsCYP3A7205 compoundsNFE2L2202 compoundsSYK201 compoundsTYROSINE-PROTEIN201 compoundsCHAIN197 compoundsGLI3194 compoundsPGR189 compoundsRATTUS188 compounds
5
A
ABCB1145ABCB1147ABCC117ABCC231ABCC315ABCC419ABCG222ABHD17B10ABHD411ABL121ACHE68ADCY915ADENOSINE23ADORA114ADORA342ADRA1A121ADRA1B41ADRA1D40ADRA2A84ADRA2B74ADRA2C76ADRB144ADRB282ADRB331AGTR113AHR89AKR1B114AKR1B1016ALB11ALDEHYDE59ALOX1228ALOX1526ALOX15B15ALOX514ALPHA-1A34ALPHA-1B33ALPHA-1D36ALPHA-2A48ALPHA-2B39ALPHA-2C34ALPI10AMINE15ANDROGEN49ANO117APAF117APOBEC3G12APP27AR296ATAD571ATG4B8ATXN272AURKB18AVPR1A11AVPR28
B
C
CA148CA1236CA1310CA1423CA244CA313CA435CA5A35CA5B34CA631CA738CA934CACNA1B9CACNA1C24CACNA1H14CAR1312CAR1519CARBONIC17CASP19CASP341CASP69CASP733CATECHOL36CBX129CDC25B9CDK116CDK512CDK5R19CFTR66CGAS15CGMP-INHIBITED21CHAIN197CHRM1130CHRM257CHRM339CHRM444CHRM545CHRNA109CHRNA411CHRNA710CHRNB210CHRNB49CIB19CISD19CLK115CNR112CREB143CSNK2A115CSNK2A212CSNK2A39CSNK2B10CTDSP18CXCL810CYCLIN-DEPENDENT11CYP19A1102CYP1A115CYP1A2230CYP1B119CYP2C19334CYP2C88CYP2C9295CYP2D6324CYP3A4224CYP3A7205CYTOCHROME244
D
E
F
G
GAA10GABRA114GABRA213GABRA313GABRA413GABRA512GABRA612GABRB112GABRB213GABRB313GABRD12GABRE12GABRG112GABRG213GABRG312GABRP12GALR312GAMMA-AMINOBUTYRIC10GAMT37GAPDH24GFER31GHSR14GLI110GLI3194GLP1R16GLRA110GLS30GLUCOCORTICOID40GLUTATHIONE21GMNN58GNAI116GNMT37GNRHR24GPBAR123GPR15129GPR3227GPR3515GPT217GPX123GPX425GRIN120GRIN2A17GRIN2B17GRIN2C16GRIN2D16GRIN3A15GRIN3B15GRK210GSK3A15GSK3B19GSTO112
H
HCRTR115HDAC111HDAC1013HDAC1112HDAC211HDAC311HDAC412HDAC512HDAC634HDAC712HDAC811HDAC940HEAT8HIF1A45HISTAMINE26HISTONE-LYSINE175HLA-B35HNF4A8HNMT37HOMO118HOXA911HPGD25HRH155HRH238HRH315HRH49HSF117HSP90AA130HSP90AB116HSPB136HSPD110HSPE110HTR1A87HTR1B32HTR1D30HTR1E20HTR1F21HTR2A117HTR2B78HTR2C61HTR3A18HTR3B11HTR49HTR5A27HTR636HTR738HTT35
I
J
K
L
M
N
O
P
PABPC112PARP116PAX826PDE4A18PDE4D25PGR189PHOSPHATIDYLINOSITOL14PHOSPHOLIPID24PIK3CG8PIM113PIM210PIP4K2A14PKM11PLA2G720PLAU9PLAUR8PLCG18PLG12PLK113PMP2267PNMT39POLB30POLH22POLI27POLK45POLY14PPARA18PPARD36PPARG83PPP1CA13PPP1R15A30PREPL8PRKAA111PRKAA213PRKAB110PRKAB210PRKAG110PRKAG210PRKAG310PRMT117PRNP10PROSTAGLANDIN14PROTEIN10PROTHROMBIN8PSIP113PSMB512PTBP111PTGER228PTGS177PTGS251PTPN115
R
S
SAE19SCN1A22SCN2A28SCN3A23SCN5A19SENP610SENP79SENP820SERPINA623SHBG35SIGMA15SIGMAR124SIRT510SLC18A211SLC22A118SLC22A119SLC22A217SLC22A39SLC22A622SLC22A826SLC29A19SLC47A115SLC5A713SLC6A264SLC6A370SLC6A467SLCO1A110SLCO1A58SLCO1B125SLCO1B319SLCO2B116SMAD249SMAD363SMARCA48SMN218SNCA23SODIUM-DEPENDENT58SRC12STK1610STK3357SUBSTANCE-K9SYK201
T
TAAR120TACR115TARDBP19TBXA2R25TDP1241TFE311THPO24THRB230THROMBOXANE-A8THYROID17TLR38TMEM9715TNFRSF10B16TOP110TOP1P137TOP2A14TP53151TRA11TRHR19TRPA123TRPC415TRPC615TRPM211TRPM78TSHR77TTR17TUBA1A9TUBA1B9TUBA1C9TUBA3C9TUBA3E9TUBA4A9TUBB9TUBB19TUBB2A9TUBB2B9TUBB39TUBB4A9TUBB4B9TUBB69TUBB89TXNRD121TYROSINE-PROTEIN201