pirenperone — Mechanism Gap Analysis
HYPOTHESIS_ENGINE_v1.0 · Corpus v20260227-01 · Deterministic graph-traversal
Known Targets
CYP2D6ESR1ESRRACYP3A7RATTUSKCNH2CHRM1DRD35-HYDROXYTRYPTAMINEHTR2ADRD2DRD1HTR1AHTR2BACHEHTR2CHTR7HTR1BGPR151S1PR4ARSA
21 known targets mapped from PubChem bioassay data
Pathway Context
Class A/1 (Rhodopsin-like receptors)10 targets overlapping
Amine ligand-binding receptors9 targets overlapping
Serotonin receptors5 targets overlapping
Uncovered Pathway Targets
159 totalADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2+149 more…
Genes present in the top pathway union that pirenperone does not directly modulate.
Top Stack Candidates
Aripiprazole
score 5,551.533#1 gap-filler · 25 targets covered · evidence score 52.0
ADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1AVPR1A+13
Fluoxetine
score 5,063.456#2 gap-filler · 16 targets covered · evidence score 73.4
ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CCCKBRCHRM3CHRM5CNR1EDNRAHRH1+4
617 more candidates · full stack optimisation locked
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BiohacksAI maps biological mechanisms. It does not recommend compounds. Results generated by HYPOTHESIS_ENGINE_v1.0.