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Compounds That Target BRD4

bromodomain containing 4 · 92 compounds in BiohacksAI corpus

BRD4 (bromodomain containing 4) is a biological target with 92 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into BRD4 modulation for therapeutic and biohacking applications.

Most Studied Compounds for BRD4
500+
studies
300+
studies
299+
studies
142+
studies
11+
studies
All 50 Compounds — Ranked by Evidence
1
Ly 294002
4.84
confidence
2
Panobinostat
4.26
confidence
3
Bi 2536
4.01
confidence
4
Romidepsin
3.95
confidence
5
Belinostat
3.91
confidence
6
Lenalidomide
3.91
confidence
7
Alprazolam
3.89
confidence
8
Dinaciclib
3.87
confidence
9
Molibresib
3.81
confidence
10
Apabetalone
3.66
confidence
11
Sb 202190
3.64
confidence
12
Birabresib
3.47
confidence
13
Fedratinib
3.40
confidence
14
Tacedinaline
3.37
confidence
15
Cloxyquin
3.04
confidence
16
Mivebresib
3.00
confidence
17
Nitroxoline
3.00
confidence
18
Volasertib
2.94
confidence
19
Abbv 744
2.56
confidence
20
Gsk046
2.40
confidence
21
Gsk620
2.30
confidence
22
Azd 5153
2.20
confidence
23
Inobrodib
2.20
confidence
24
Ischemin
2.20
confidence
25
Methylpyrrolidone
2.20
confidence
26
Gsk778
2.08
confidence
27
Withanolide E
1.95
confidence
28
35 Dimethyl 4 Phenylisoxazole
1.79
confidence
29
Agastache Rugosa
1.00
confidence
30
Artemisia Annua
1.00
confidence
31
Bupleurum Chinense
1.00
confidence
32
Fritillaria Cirrhosa
1.00
confidence
299+
studies
1.00
confidence
1.00
confidence
300+
studies
1.00
confidence
36
Prunus Mume
1.00
confidence
37
Rehmannia Glutinosa
1.00
confidence
38
Sargassum Fusiforme
1.00
confidence
39
Scutellaria Baicalensis
1.00
confidence
142+
studies
1.00
confidence
41
Ziziphus Jujuba
1.00
confidence
11+
studies
0.69
confidence
2+
studies
0.69
confidence
2+
studies
0.69
confidence
2+
studies
0.69
confidence
46
Achyranthes Bidentata
0.50
confidence
500+
studies
0.50
confidence
48
Aloe Vera
0.50
confidence
49
Anemarrhena Asphodeloides
0.50
confidence
50
Arctium Lappa
0.50
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for BRD4 (bromodomain containing 4). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: BRD4 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.