BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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Compounds That Target CXCR4

C-X-C chemokine receptor type 4 · 124 compounds in BiohacksAI corpus

CXCR4 (C-X-C chemokine receptor type 4) is a biological target with 124 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into CXCR4 modulation for therapeutic and biohacking applications.

Most Studied Compounds for CXCR4
500+
studies
500+
studies
500+
studies
500+
studies
499+
studies
300+
studies
299+
studies
All 51 Compounds — Ranked by Evidence
1
Plerixafor
4.20
confidence
2
Mavorixafor
2.77
confidence
500+
studies
1.00
confidence
4
Allium Tuberosum
1.00
confidence
5
Aloe Vera
1.00
confidence
6
Anemarrhena Asphodeloides
1.00
confidence
7
Apis Mellifera
1.00
confidence
8
Arctium Lappa
1.00
confidence
9
Artemisia Annua
1.00
confidence
10
Artemisia Argyi
1.00
confidence
11
Artemisia Capillaris
1.00
confidence
12
Aster Tataricus
1.00
confidence
13
Atractylodes Macrocephala
1.00
confidence
14
Bombyx Mori
1.00
confidence
15
Bufo Bufo
1.00
confidence
16
Bupleurum Chinense
1.00
confidence
499+
studies
1.00
confidence
18
Chaenomeles Speciosa
1.00
confidence
19
Citrus Reticulata
1.00
confidence
500+
studies
1.00
confidence
21
Cuscuta Chinensis
1.00
confidence
22
Cynomorium Songaricum
1.00
confidence
23
Ephedra Sinica
1.00
confidence
24
Eriobotrya Japonica
1.00
confidence
25
Eucommia Ulmoides
1.00
confidence
26
Forsythia Suspensa
1.00
confidence
27
Fritillaria Cirrhosa
1.00
confidence
28
Gastrodia Elata
1.00
confidence
299+
studies
1.00
confidence
30
Glycine Max
1.00
confidence
31
Glycyrrhiza Uralensis
1.00
confidence
32
Lilium Lancifolium
1.00
confidence
33
Litchi Chinensis
1.00
confidence
34
Lithospermum Erythrorhizon
1.00
confidence
35
Lobelia Chinensis
1.00
confidence
36
Lonicera Japonica
1.00
confidence
37
Morus Alba
1.00
confidence
1.00
confidence
39
Paeonia Lactiflora
1.00
confidence
300+
studies
1.00
confidence
41
Panax Notoginseng
1.00
confidence
42
Perilla Frutescens
1.00
confidence
43
Pinellia Ternata
1.00
confidence
44
Polygala Tenuifolia
1.00
confidence
45
Polygonum Cuspidatum
1.00
confidence
500+
studies
1.00
confidence
47
Prunus Armeniaca
1.00
confidence
48
Prunus Mume
1.00
confidence
500+
studies
1.00
confidence
50
Agastache Rugosa
1.00
confidence
2+
studies
0.69
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for CXCR4 (C-X-C chemokine receptor type 4). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: CXCR4 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.