BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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Compounds That Target CYP2B6

cytochrome P450 family 2 subfamily B member 6 · 125 compounds in BiohacksAI corpus

CYP2B6 (cytochrome P450 family 2 subfamily B member 6) is a cytochrome P450 enzyme involved in the metabolism of drugs, hormones, and dietary compounds. CYP enzymes are critical determinants of pharmacokinetics and drug-herb interactions. The 125 compounds listed here have documented interactions with CYP2B6 based on BindingDB inhibition and binding assay data, making this resource valuable for assessing compound safety and interaction profiles.

Most Studied Compounds for CYP2B6
500+
studies
500+
studies
500+
studies
499+
studies
499+
studies
300+
studies
300+
studies
299+
studies
299+
studies
298+
studies
All 53 Compounds — Ranked by Evidence
1
Tranylcypromine
4.48
confidence
299+
studies
2.20
confidence
300+
studies
1.10
confidence
500+
studies
1.00
confidence
1.00
confidence
6
Polygala Tenuifolia
1.00
confidence
7
Polygonum Cuspidatum
1.00
confidence
8
Achyranthes Bidentata
1.00
confidence
9
Agastache Rugosa
1.00
confidence
500+
studies
1.00
confidence
11
Allium Tuberosum
1.00
confidence
12
Aloe Vera
1.00
confidence
13
Arctium Lappa
1.00
confidence
14
Artemisia Annua
1.00
confidence
15
Artemisia Argyi
1.00
confidence
16
Artemisia Capillaris
1.00
confidence
17
Aster Tataricus
1.00
confidence
18
Atractylodes Macrocephala
1.00
confidence
19
Bombyx Mori
1.00
confidence
20
Carthamus Tinctorius
1.00
confidence
499+
studies
1.00
confidence
22
Chaenomeles Speciosa
1.00
confidence
23
Citrus Reticulata
1.00
confidence
24
Commiphora Myrrha
1.00
confidence
25
Crataegus Pinnatifida
1.00
confidence
500+
studies
1.00
confidence
27
Cuscuta Chinensis
1.00
confidence
28
Dimocarpus Longan
1.00
confidence
29
Ephedra Sinica
1.00
confidence
30
Eriobotrya Japonica
1.00
confidence
31
Eucommia Ulmoides
1.00
confidence
499+
studies
1.00
confidence
33
Forsythia Suspensa
1.00
confidence
34
Fritillaria Cirrhosa
1.00
confidence
35
Gastrodia Elata
1.00
confidence
36
Gentiana Macrophylla
1.00
confidence
299+
studies
1.00
confidence
38
Glycine Max
1.00
confidence
39
Glycyrrhiza Uralensis
1.00
confidence
40
Lilium Lancifolium
1.00
confidence
41
Litchi Chinensis
1.00
confidence
42
Lithospermum Erythrorhizon
1.00
confidence
43
Lonicera Japonica
1.00
confidence
44
Morus Alba
1.00
confidence
1.00
confidence
46
Paeonia Lactiflora
1.00
confidence
300+
studies
1.00
confidence
48
Panax Notoginseng
1.00
confidence
49
Perilla Frutescens
1.00
confidence
50
Pinellia Ternata
1.00
confidence
298+
studies
0.69
confidence
296+
studies
0.69
confidence
53
298+
studies
0.69
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for CYP2B6 (cytochrome P450 family 2 subfamily B member 6). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: CYP2B6 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.