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Compounds That Target DDR1

discoidin domain receptor tyrosine kinase 1 · 68 compounds in BiohacksAI corpus

DDR1 (discoidin domain receptor tyrosine kinase 1) is a biological target with 68 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into DDR1 modulation for therapeutic and biohacking applications.

All 50 Compounds — Ranked by Evidence
1
Erlotinib
5.55
confidence
2
Imatinib
5.47
confidence
3
Sb 203580
4.92
confidence
4
Cabozantinib
4.39
confidence
5
Foretinib
4.34
confidence
6
Tozasertib
4.33
confidence
7
Vandetanib
4.30
confidence
8
Ponatinib
4.26
confidence
9
Nilotinib
4.17
confidence
10
Bosutinib
4.08
confidence
11
Doramapimod
4.06
confidence
12
Quizartinib
3.99
confidence
13
Midostaurin
3.85
confidence
14
Pazopanib
3.69
confidence
15
Vatalanib
3.69
confidence
16
Sb 202190
3.64
confidence
17
Nintedanib
3.61
confidence
18
Regorafenib
3.56
confidence
19
Canertinib
3.53
confidence
20
Tae 684
3.43
confidence
21
Fedratinib
3.40
confidence
22
Bms 777607
3.37
confidence
23
Linifanib
3.33
confidence
24
Mln 8054
3.33
confidence
25
Saracatinib
3.33
confidence
26
Neflamapimod
3.30
confidence
27
Tandutinib
3.22
confidence
28
Dovitinib
3.09
confidence
29
Dasatinib Anhydrous
3.09
confidence
30
Lestaurtinib
3.04
confidence
31
Pacritinib
3.04
confidence
32
Lenvatinib
3.04
confidence
33
Danusertib
2.94
confidence
34
Defosbarasertib
2.89
confidence
35
R 406
2.83
confidence
36
Cediranib
2.83
confidence
37
Milciclib
2.77
confidence
38
Masitinib
2.77
confidence
39
Pha 665752
2.71
confidence
40
Plx 4720
2.71
confidence
41
Enmd 2076
2.71
confidence
42
Kw 2449
2.64
confidence
43
Tivozanib
2.64
confidence
44
Bemcentinib
2.64
confidence
45
Ast 487
2.56
confidence
46
Raf 265
2.48
confidence
47
Motesanib
2.48
confidence
48
Brivanib
2.48
confidence
49
Mk 5108
2.48
confidence
50
Merestinib
2.48
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for DDR1 (discoidin domain receptor tyrosine kinase 1). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: DDR1 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.