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Compounds That Target GRK1

Rhodopsin kinase GRK1 · 86 compounds in BiohacksAI corpus

GRK1 (Rhodopsin kinase GRK1) is a receptor that mediates ligand-dependent signaling relevant to physiology, behavior, and metabolism. The 86 compounds with documented GRK1 interactions span synthetic agonists, antagonists, and natural ligands identified through BindingDB binding assays and PubMed literature in the BiohacksAI corpus.

Most Studied Compounds for GRK1
500+
studies
500+
studies
300+
studies
299+
studies
199+
studies
All 50 Compounds — Ranked by Evidence
1
Alvocidib
4.52
confidence
2
Ruxolitinib
4.23
confidence
3
Midostaurin
3.85
confidence
4
Nintedanib
3.61
confidence
5
Tae 684
3.43
confidence
6
Dovitinib
3.09
confidence
7
Lestaurtinib
3.04
confidence
8
Sangivamycin
3.00
confidence
9
Ruboxistaurin
2.94
confidence
10
R 406
2.83
confidence
11
Pha 665752
2.71
confidence
12
Gsk 690693
2.64
confidence
13
Balanol
2.30
confidence
14
Su 014813
2.20
confidence
15
Enzastaurin
2.08
confidence
16
Aloe Vera
1.00
confidence
17
Artemisia Argyi
1.00
confidence
18
Artemisia Capillaris
1.00
confidence
19
Carthamus Tinctorius
1.00
confidence
20
Citrus Reticulata
1.00
confidence
500+
studies
1.00
confidence
22
Ephedra Sinica
1.00
confidence
299+
studies
1.00
confidence
24
Lobelia Chinensis
1.00
confidence
25
Lonicera Japonica
1.00
confidence
1.00
confidence
300+
studies
1.00
confidence
28
Panax Notoginseng
1.00
confidence
29
Prunus Armeniaca
1.00
confidence
30
Prunus Mume
1.00
confidence
31
Quisqualis Indica
1.00
confidence
500+
studies
1.00
confidence
33
Rehmannia Glutinosa
1.00
confidence
34
Trichosanthes Kirilowii
1.00
confidence
498+
studies
1.00
confidence
36
Achyranthes Bidentata
0.50
confidence
37
Aconitum Carmichaelii
0.50
confidence
38
Allium Fistulosum
0.50
confidence
39
Allium Tuberosum
0.50
confidence
40
Apis Mellifera
0.50
confidence
41
Aquilaria Sinensis
0.50
confidence
42
Arctium Lappa
0.50
confidence
199+
studies
0.50
confidence
44
Asparagus Cochinchinensis
0.50
confidence
45
Aucklandia Lappa
0.50
confidence
46
Belamcanda Chinensis
0.50
confidence
47
Bupleurum Chinense
0.50
confidence
48
Chaenomeles Speciosa
0.50
confidence
49
Cimicifuga Heracleifolia
0.50
confidence
50
Cnidium Monnieri
0.50
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for GRK1 (Rhodopsin kinase GRK1). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: GRK1 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.