BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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Compounds That Target GRK5

G protein-coupled receptor kinase 5 · 111 compounds in BiohacksAI corpus

GRK5 (G protein-coupled receptor kinase 5) is a receptor that mediates ligand-dependent signaling relevant to physiology, behavior, and metabolism. The 111 compounds with documented GRK5 interactions span synthetic agonists, antagonists, and natural ligands identified through BindingDB binding assays and PubMed literature in the BiohacksAI corpus.

Most Studied Compounds for GRK5
500+
studies
500+
studies
500+
studies
499+
studies
300+
studies
299+
studies
142+
studies
96+
studies
All 51 Compounds — Ranked by Evidence
1
Upadacitinib
3.09
confidence
2
Balanol
2.30
confidence
3
Gsk 180736a
2.08
confidence
4
Aloe Vera
1.00
confidence
5
Apis Mellifera
1.00
confidence
6
Artemisia Capillaris
1.00
confidence
7
Aster Tataricus
1.00
confidence
8
Atractylodes Macrocephala
1.00
confidence
9
Bufo Bufo
1.00
confidence
10
Bupleurum Chinense
1.00
confidence
11
Carthamus Tinctorius
1.00
confidence
499+
studies
1.00
confidence
13
Chaenomeles Speciosa
1.00
confidence
14
Citrus Reticulata
1.00
confidence
500+
studies
1.00
confidence
16
Cuscuta Chinensis
1.00
confidence
17
Cynomorium Songaricum
1.00
confidence
18
Ephedra Sinica
1.00
confidence
19
Eriobotrya Japonica
1.00
confidence
20
Forsythia Suspensa
1.00
confidence
21
Gastrodia Elata
1.00
confidence
299+
studies
1.00
confidence
23
Ligusticum Chuanxiong
1.00
confidence
24
Litchi Chinensis
1.00
confidence
25
Lithospermum Erythrorhizon
1.00
confidence
26
Lonicera Japonica
1.00
confidence
27
Morus Alba
1.00
confidence
1.00
confidence
29
Paeonia Lactiflora
1.00
confidence
300+
studies
1.00
confidence
31
Panax Notoginseng
1.00
confidence
32
Perilla Frutescens
1.00
confidence
33
Pinellia Ternata
1.00
confidence
1.00
confidence
35
Polygala Tenuifolia
1.00
confidence
500+
studies
1.00
confidence
37
Prunus Armeniaca
1.00
confidence
38
Prunus Persica
1.00
confidence
500+
studies
1.00
confidence
40
Rehmannia Glutinosa
1.00
confidence
41
Salvia Miltiorrhiza
1.00
confidence
42
Scrophularia Ningpoensis
1.00
confidence
43
Scutellaria Baicalensis
1.00
confidence
142+
studies
1.00
confidence
45
Smilax Glabra
1.00
confidence
500+
studies
1.00
confidence
47
Trichosanthes Kirilowii
1.00
confidence
498+
studies
1.00
confidence
49
Agastache Rugosa
1.00
confidence
50
Allium Tuberosum
1.00
confidence
96+
studies
0.69
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for GRK5 (G protein-coupled receptor kinase 5). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: GRK5 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.