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Compounds That Target KCNH2

potassium voltage-gated channel subfamily H member 2 · 393 compounds in BiohacksAI corpus

KCNH2 (potassium voltage-gated channel subfamily H member 2) is a biological target with 393 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into KCNH2 modulation for therapeutic and biohacking applications.

Most Studied Compounds for KCNH2
280+
studies
All 50 Compounds — Ranked by Evidence
1
Tacrine
6.08
confidence
2
Tamoxifen
5.88
confidence
3
Clozapine
5.81
confidence
4
Imipramine
5.69
confidence
5
Nifedipine
5.34
confidence
6
Desipramine
5.23
confidence
7
Prazosin
5.15
confidence
8
Osimertinib
5.03
confidence
9
Mefloquine
4.93
confidence
10
Risperidone
4.89
confidence
11
Ibrutinib
4.86
confidence
12
Amsacrine
4.82
confidence
13
Sildenafil
4.78
confidence
14
Diltiazem
4.74
confidence
15
Lopinavir
4.64
confidence
16
Berberine Chloride
4.56
confidence
17
Terfenadine
4.55
confidence
18
Propafenone
4.53
confidence
19
Thioridazine
4.52
confidence
20
Amiodarone
4.51
confidence
21
Olanzapine
4.44
confidence
22
Paroxetine
4.39
confidence
23
Citalopram
4.36
confidence
24
Sr Mefloquine
4.28
confidence
25
Ponatinib
4.26
confidence
26
Mibefradil
4.26
confidence
27
Trifluoperazine
4.25
confidence
28
Diphenhydramine
4.22
confidence
29
Rilpivirine
4.20
confidence
30
Ceritinib
4.19
confidence
31
Pimozide
4.19
confidence
32
Nilotinib
4.17
confidence
33
Pyrilamine
4.17
confidence
34
Vanoxerine
4.08
confidence
35
Ziprasidone
3.99
confidence
36
Acacetin
3.99
confidence
37
Mexiletine
3.99
confidence
38
Ifenprodil
3.95
confidence
39
Disopyramide
3.95
confidence
40
Bupropion
3.93
confidence
41
Tadalafil
3.93
confidence
42
Fluphenazine
3.91
confidence
43
Terazosin
3.83
confidence
44
Fexofenadine
3.83
confidence
45
Atomoxetine
3.71
confidence
46
Carfilzomib
3.69
confidence
47
Abemaciclib
3.66
confidence
48
Fasudil
3.66
confidence
280+
studies
3.64
confidence
50
Nintedanib
3.61
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for KCNH2 (potassium voltage-gated channel subfamily H member 2). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: KCNH2 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.