BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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Compounds That Target MAP2K5

mitogen-activated protein kinase kinase 5 · 64 compounds in BiohacksAI corpus

MAP2K5 (mitogen-activated protein kinase kinase 5) is a biological target with 64 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into MAP2K5 modulation for therapeutic and biohacking applications.

All 50 Compounds — Ranked by Evidence
1
Gefitinib
5.67
confidence
2
Erlotinib
5.55
confidence
3
Sb 203580
4.92
confidence
4
Ibrutinib
4.86
confidence
5
Lapatinib
4.84
confidence
6
Alvocidib
4.52
confidence
7
Cabozantinib
4.39
confidence
8
Foretinib
4.34
confidence
9
Tozasertib
4.33
confidence
10
Vandetanib
4.30
confidence
11
Ponatinib
4.26
confidence
12
Nilotinib
4.17
confidence
13
Bosutinib
4.08
confidence
14
Pazopanib
3.69
confidence
15
Neratinib
3.66
confidence
16
Nintedanib
3.61
confidence
17
Canertinib
3.53
confidence
18
Tae 684
3.43
confidence
19
Fedratinib
3.40
confidence
20
Gilteritinib
3.40
confidence
21
Bms 777607
3.37
confidence
22
Linifanib
3.33
confidence
23
Dabrafenib
3.30
confidence
24
Tandutinib
3.22
confidence
25
Mirdametinib
3.18
confidence
26
Dovitinib
3.09
confidence
27
At 9283
3.09
confidence
28
Lestaurtinib
3.04
confidence
29
Lenvatinib
3.04
confidence
30
Ruboxistaurin
2.94
confidence
31
Defosbarasertib
2.89
confidence
32
Orantinib
2.89
confidence
33
Barasertib
2.89
confidence
34
R 406
2.83
confidence
35
K 252a
2.83
confidence
36
Cediranib
2.83
confidence
37
Pha 665752
2.71
confidence
38
Plx 4720
2.71
confidence
39
Crenolanib
2.71
confidence
40
Apitolisib
2.71
confidence
41
Kw 2449
2.64
confidence
42
Linsitinib
2.64
confidence
43
Ast 487
2.56
confidence
44
Cp 724714
2.56
confidence
45
Raf 265
2.48
confidence
46
Brivanib
2.48
confidence
47
Tak 285
2.40
confidence
48
Azd 7762
2.30
confidence
49
Aee 788
2.30
confidence
50
Avutometinib
2.30
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for MAP2K5 (mitogen-activated protein kinase kinase 5). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: MAP2K5 target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.