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B
MOLECULAR TARGETUniProt: O14976

GAK

cyclin G associated kinase

73 compounds · BiohacksAI corpus v20260307-01

73
compounds
Compounds
73
Gene Symbol
GAK
NCBI Gene
2580

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About GAK

GAK (cyclin G associated kinase) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 73 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View GAK on UniProt →
Compounds Targeting GAK (50)
1
Gefitinib
5.67
confidence
2
Erlotinib
5.55
confidence
3
Imatinib
5.47
confidence
4
Sb 203580
4.92
confidence
5
Alvocidib
4.52
confidence
6
Tozasertib
4.33
confidence
7
Vandetanib
4.30
confidence
8
Ponatinib
4.26
confidence
9
Ruxolitinib
4.23
confidence
10
Bosutinib
4.08
confidence
11
Bi 2536
4.01
confidence
12
Midostaurin
3.85
confidence
13
Silmitasertib
3.78
confidence
14
Pazopanib
3.69
confidence
15
Neratinib
3.66
confidence
16
Abemaciclib
3.66
confidence
17
Sb 202190
3.64
confidence
18
Baricitinib
3.56
confidence
19
Canertinib
3.53
confidence
20
Pelitinib
3.50
confidence
21
Bms 387032
3.47
confidence
22
Tae 684
3.43
confidence
23
Fedratinib
3.40
confidence
24
Gilteritinib
3.40
confidence
25
Linifanib
3.33
confidence
26
Saracatinib
3.33
confidence
27
Sgi 1776
3.26
confidence
28
Ribociclib
3.26
confidence
29
Tandutinib
3.22
confidence
30
Sp 600125
3.22
confidence
31
Alectinib
3.18
confidence
32
Rociletinib
3.18
confidence
33
Dacomitinib Anhydrous
3.14
confidence
34
Dovitinib
3.09
confidence
35
Jnj 7706621
3.09
confidence
36
At 9283
3.09
confidence
37
Upadacitinib
3.09
confidence
38
Lestaurtinib
3.04
confidence
39
Pacritinib
3.04
confidence
40
Adavosertib
3.04
confidence
41
Pf 03758309
3.00
confidence
42
Ruboxistaurin
2.94
confidence
43
Galunisertib
2.94
confidence
44
Momelotinib
2.89
confidence
45
Orantinib
2.89
confidence
46
R 406
2.83
confidence
47
K 252a
2.83
confidence
48
Cediranib
2.83
confidence
49
Milciclib
2.77
confidence
50
Pha 665752
2.71
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.