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Compounds That Target ADORA2A

adenosine A2a receptor · 94 compounds in BiohacksAI corpus

ADORA2A (adenosine A2a receptor) is a biological target with 94 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into ADORA2A modulation for therapeutic and biohacking applications.

Most Studied Compounds for ADORA2A
500+
studies
300+
studies
300+
studies
300+
studies
299+
studies
298+
studies
All 50 Compounds — Ranked by Evidence
1
Tamoxifen
5.88
confidence
2
Nifedipine
5.34
confidence
3
Allopurinol
5.04
confidence
4
Sb 203580
4.92
confidence
5
Neca
4.86
confidence
6
Sildenafil
4.78
confidence
7
Raloxifene
4.77
confidence
8
13 Dipropyl 8 Cyclopentylxanthine Dpcpx
4.57
confidence
9
Galangin
4.30
confidence
10
N6 Cyclopentyladenosine
4.28
confidence
11
Sr Mefloquine
4.28
confidence
12
Diethylstilbestrol
4.06
confidence
13
Gentian Violet
4.03
confidence
14
Ib Meca
4.01
confidence
15
Amiloride
3.95
confidence
16
Namodenoson
3.95
confidence
17
Zm 241385
3.87
confidence
18
Cgs 21680
3.66
confidence
19
S Dhpa
3.64
confidence
20
Istradefylline
3.50
confidence
21
Cgs 15943
3.47
confidence
22
R Pia
3.47
confidence
23
Sch 58261
3.40
confidence
24
Xanthine Amine Congener
3.37
confidence
25
8 Phenyl Theophylline
3.26
confidence
26
Imiquimod
3.14
confidence
27
Enprofylline
2.94
confidence
300+
studies
2.89
confidence
29
Bithionol
2.89
confidence
30
Psilocin
2.77
confidence
31
Rolofylline
2.71
confidence
32
Nn Hexamethyleneamiloride
2.56
confidence
33
Defactinib
2.48
confidence
34
Gsk046
2.40
confidence
35
S Pia
2.40
confidence
36
Trioxsalen
2.30
confidence
298+
studies
2.20
confidence
38
Regadenoson Anhydrous
2.20
confidence
39
Metrifudil
2.20
confidence
40
Tozadenant
2.08
confidence
41
Ciforadenant
1.95
confidence
42
Tecadenoson
1.95
confidence
299+
studies
1.79
confidence
44
Rs Mefloquine
1.79
confidence
45
St1535
1.79
confidence
46
Binodenoson
1.79
confidence
47
Glycyrrhiza Uralensis
1.00
confidence
300+
studies
0.69
confidence
300+
studies
0.69
confidence
500+
studies
0.50
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for ADORA2A (adenosine A2a receptor). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: ADORA2A target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.