BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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Compounds That Target AR

androgen receptor · 436 compounds in BiohacksAI corpus

AR (androgen receptor) is a receptor that mediates ligand-dependent signaling relevant to physiology, behavior, and metabolism. The 436 compounds with documented AR interactions span synthetic agonists, antagonists, and natural ligands identified through BindingDB binding assays and PubMed literature in the BiohacksAI corpus.

Most Studied Compounds for AR
1.0k+
studies
1.0k+
studies
300+
studies
300+
studies
300+
studies
300+
studies
300+
studies
300+
studies
All 50 Compounds — Ranked by Evidence
1
Dorzolamide
4.86
confidence
300+
studies
4.62
confidence
3
Enzalutamide
4.61
confidence
4
Stanolone
4.55
confidence
5
Gossypol
4.42
confidence
299+
studies
3.66
confidence
7
R Bicalutamide
3.53
confidence
299+
studies
3.53
confidence
299+
studies
3.37
confidence
298+
studies
3.33
confidence
11
5 Hydroxyflavone
3.33
confidence
298+
studies
3.30
confidence
13
Metribolone
3.30
confidence
300+
studies
3.18
confidence
292+
studies
3.18
confidence
16
Tolfenamic Acid
3.09
confidence
300+
studies
3.04
confidence
18
Tiratricol
3.04
confidence
300+
studies
3.00
confidence
300+
studies
3.00
confidence
1.0k+
studies
2.94
confidence
300+
studies
2.89
confidence
23
Guggulsterone
2.89
confidence
299+
studies
2.83
confidence
1.0k+
studies
2.83
confidence
300+
studies
2.83
confidence
298+
studies
2.83
confidence
298+
studies
2.83
confidence
29
Bufalin
2.83
confidence
300+
studies
2.77
confidence
300+
studies
2.77
confidence
298+
studies
2.77
confidence
278+
studies
2.71
confidence
34
2 Hydroxy Flavanone
2.71
confidence
35
Bisphenol A
2.71
confidence
119+
studies
2.71
confidence
300+
studies
2.71
confidence
38
Nandrolonepolycyclic
2.64
confidence
39
Galeterone
2.64
confidence
300+
studies
2.56
confidence
300+
studies
2.56
confidence
300+
studies
2.56
confidence
299+
studies
2.48
confidence
299+
studies
2.48
confidence
299+
studies
2.48
confidence
300+
studies
2.48
confidence
300+
studies
2.48
confidence
297+
studies
2.48
confidence
300+
studies
2.48
confidence
298+
studies
2.48
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for AR (androgen receptor). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: AR target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.