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Compounds That Target CIT

citron rho-interacting serine/threonine kinase · 140 compounds in BiohacksAI corpus

CIT (citron rho-interacting serine/threonine kinase) is a biological target with 140 documented compound interactions in the BiohacksAI corpus. The compounds listed below have been identified through computational analysis of BindingDB binding assay data and PubMed literature. Each interaction is ranked by confidence score reflecting the breadth and strength of experimental evidence. This resource supports research into CIT modulation for therapeutic and biohacking applications.

Most Studied Compounds for CIT
500+
studies
300+
studies
299+
studies
297+
studies
11+
studies
All 52 Compounds — Ranked by Evidence
1
Gefitinib
5.67
confidence
2
Erlotinib
5.55
confidence
3
Sb 203580
4.92
confidence
4
Alvocidib
4.52
confidence
5
Foretinib
4.34
confidence
6
Vandetanib
4.30
confidence
7
Ruxolitinib
4.23
confidence
8
Bosutinib
4.08
confidence
9
Doramapimod
4.06
confidence
10
Bi 2536
4.01
confidence
11
Vatalanib
3.69
confidence
12
Abemaciclib
3.66
confidence
13
Fasudil
3.66
confidence
14
Sb 202190
3.64
confidence
15
Baricitinib
3.56
confidence
16
Canertinib
3.53
confidence
17
Pelitinib
3.50
confidence
18
Bms 387032
3.47
confidence
19
Gilteritinib
3.40
confidence
20
Fedratinib
3.40
confidence
21
Dovitinib
3.09
confidence
22
Lestaurtinib
3.04
confidence
23
Ruboxistaurin
2.94
confidence
24
Momelotinib
2.89
confidence
25
Defosbarasertib
2.89
confidence
26
R 406
2.83
confidence
27
Kw 2449
2.64
confidence
28
Gsk 690693
2.64
confidence
29
Ast 487
2.56
confidence
30
Raf 265
2.48
confidence
31
Motesanib
2.48
confidence
32
Su 014813
2.20
confidence
33
Y 39983
2.20
confidence
34
Gsk 1070916
2.20
confidence
35
Cyc 116
2.08
confidence
36
Afuresertib
1.79
confidence
300+
studies
1.39
confidence
299+
studies
1.00
confidence
39
Forsythia Suspensa
1.00
confidence
40
Gastrodia Elata
1.00
confidence
41
Allium Tuberosum
1.00
confidence
42
Artemisia Argyi
1.00
confidence
43
Artemisia Capillaris
1.00
confidence
44
Aster Tataricus
1.00
confidence
45
Atractylodes Macrocephala
1.00
confidence
46
Chaenomeles Speciosa
1.00
confidence
47
Citrus Reticulata
1.00
confidence
500+
studies
1.00
confidence
49
Ephedra Sinica
1.00
confidence
50
Eriobotrya Japonica
1.00
confidence
297+
studies
0.69
confidence
11+
studies
0.69
confidence

The compounds above were identified through computational analysis of BindingDB binding assay data and PubMed literature for CIT (citron rho-interacting serine/threonine kinase). Confidence scores reflect the strength and breadth of experimental evidence.

Explore related resources: CIT target overview · All biological targets · Biological pathways

Data from BindingDB and PubMed. For research purposes only. Not medical advice.