BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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B
MOLECULAR TARGETUniProt: O14578

CIT

citron rho-interacting serine/threonine kinase

39 compounds · BiohacksAI corpus v20260307-01

39
compounds
Compounds
39
Gene Symbol
CIT
NCBI Gene
11113

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About CIT

CIT (citron rho-interacting serine/threonine kinase) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 39 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View CIT on UniProt →
Compounds Targeting CIT (39)
1
Gefitinib
5.67
confidence
2
Erlotinib
5.55
confidence
3
Sb 203580
4.92
confidence
4
Alvocidib
4.52
confidence
5
Foretinib
4.34
confidence
6
Vandetanib
4.30
confidence
7
Ruxolitinib
4.23
confidence
8
Bosutinib
4.08
confidence
9
Doramapimod
4.06
confidence
10
Bi 2536
4.01
confidence
11
Vatalanib
3.69
confidence
12
Abemaciclib
3.66
confidence
13
Fasudil
3.66
confidence
14
Sb 202190
3.64
confidence
15
Baricitinib
3.56
confidence
16
Canertinib
3.53
confidence
17
Pelitinib
3.50
confidence
18
Bms 387032
3.47
confidence
19
Fedratinib
3.40
confidence
20
Gilteritinib
3.40
confidence
21
Dovitinib
3.09
confidence
22
Lestaurtinib
3.04
confidence
23
Ruboxistaurin
2.94
confidence
24
Defosbarasertib
2.89
confidence
25
Momelotinib
2.89
confidence
26
R 406
2.83
confidence
27
Kw 2449
2.64
confidence
28
Gsk 690693
2.64
confidence
29
Ast 487
2.56
confidence
30
Raf 265
2.48
confidence
31
Motesanib
2.48
confidence
32
Su 014813
2.20
confidence
33
Gsk 1070916
2.20
confidence
34
Y 39983
2.20
confidence
35
Cyc 116
2.08
confidence
36
Afuresertib
1.79
confidence
300
studies
1.39
confidence
297
studies
0.69
confidence
11
studies
0.69
confidence
Top 39 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.