MOLECULAR TARGETUniProt: Q06187
BTK
Bruton tyrosine kinase
50 compounds · BiohacksAI corpus v20260307-01
50
compounds
Compounds
50
Gene Symbol
BTK
NCBI Gene
695
Looking for compounds that interact with BTK?
View all 50 compounds →About BTK
BTK (Bruton tyrosine kinase) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 50 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.
View BTK on UniProt →Compounds Targeting BTK (50)
1
Osimertinib
5.03
confidence
2
Ibrutinib
4.86
confidence
3
Foretinib
4.34
confidence
4
Tozasertib
4.33
confidence
5
Vandetanib
4.30
confidence
6
Ponatinib
4.26
confidence
7
Ceritinib
4.19
confidence
8
Bosutinib
4.08
confidence
9
Brigatinib
3.81
confidence
10
Neratinib
3.66
confidence
11
Nintedanib
3.61
confidence
12
Canertinib
3.53
confidence
13
Pelitinib
3.50
confidence
14
Tae 684
3.43
confidence
15
Fedratinib
3.40
confidence
16
Mln 8054
3.33
confidence
17
Saracatinib
3.33
confidence
18
Acalabrutinib
3.22
confidence
19
Rociletinib
3.18
confidence
20
Sulfuretin
3.14
confidence
21
At 9283
3.09
confidence
22
Lestaurtinib
3.04
confidence
23
Spebrutinib
3.04
confidence
24
Pf 03758309
3.00
confidence
25
Danusertib
2.94
confidence
26
Defosbarasertib
2.89
confidence
27
R 406
2.83
confidence
28
K 252a
2.83
confidence
29
Cediranib
2.83
confidence
30
Ritlecitinib
2.77
confidence
31
Apitolisib
2.71
confidence
32
Kw 2449
2.64
confidence
33
Zanubrutinib
2.56
confidence
34
Poziotinib
2.48
confidence
35
Evobrutinib
2.48
confidence
36
Entospletinib
2.48
confidence
37
Azd 7762
2.30
confidence
38
Bms 754807
2.30
confidence
39
Olmutinib
2.30
confidence
40
Su 014813
2.20
confidence
41
Rebastinib
2.20
confidence
42
Futibatinib
2.20
confidence
43
Asp 3026
2.08
confidence
44
Tirabrutinib
1.95
confidence
45
Ucn 01
1.79
confidence
46
Tolebrutinib
1.79
confidence
298
studies
0.69
confidence
299
studies
0.69
confidence
4
studies
0.69
confidence
2
studies
0.69
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed
All data is computationally derived from published research. Not medical advice. Independent validation required.