BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
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B
MOLECULAR TARGETUniProt: P04626

ERBB2

erb-b2 receptor tyrosine kinase 2

74 compounds · BiohacksAI corpus v20260307-01

74
compounds
Compounds
74
Gene Symbol
ERBB2
NCBI Gene
2064

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About ERBB2

ERBB2 (erb-b2 receptor tyrosine kinase 2) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 74 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View ERBB2 on UniProt →
Compounds Targeting ERBB2 (50)
1
Paclitaxel
7.17
confidence
2
Tamoxifen
5.88
confidence
3
Gefitinib
5.67
confidence
4
Erlotinib
5.55
confidence
5
Imatinib
5.47
confidence
6
Osimertinib
5.03
confidence
7
Sb 203580
4.92
confidence
8
Ibrutinib
4.86
confidence
9
Lapatinib
4.84
confidence
10
Alvocidib
4.52
confidence
11
Amiodarone
4.51
confidence
12
Foretinib
4.34
confidence
13
Vandetanib
4.30
confidence
14
Caffeic Acid Phenethyl Ester
4.25
confidence
15
Bosutinib
4.08
confidence
16
Fluphenazine
3.91
confidence
17
Brigatinib
3.81
confidence
18
Neratinib
3.66
confidence
19
Canertinib
3.53
confidence
20
Pelitinib
3.50
confidence
21
Candesartan
3.47
confidence
22
Tae 684
3.43
confidence
23
Acalabrutinib
3.22
confidence
24
Dacomitinib Anhydrous
3.14
confidence
25
Defosbarasertib
2.89
confidence
26
Bithionol
2.89
confidence
27
Pu H71
2.89
confidence
28
Benzodefchrysene
2.89
confidence
29
Cediranib
2.83
confidence
30
Masitinib
2.77
confidence
31
Closantel
2.71
confidence
32
Ebastine
2.64
confidence
33
Zanubrutinib
2.56
confidence
34
Cp 724714
2.56
confidence
35
Poziotinib
2.48
confidence
36
Tyrphostin 47
2.48
confidence
37
Cudc 101
2.40
confidence
38
Benzethonium Chloride
2.40
confidence
39
Tak 285
2.40
confidence
40
Aee 788
2.30
confidence
41
Cetylpyridinium Bromide
2.20
confidence
42
Iodoquinol
2.20
confidence
43
Mubritinib
2.20
confidence
44
Tg100 115
2.08
confidence
45
Enclomiphene
2.08
confidence
46
Canertinib Dihydrochloride
2.08
confidence
47
Lapatinib Ditosylate
2.08
confidence
48
Tyrphostin Ag 879
2.08
confidence
49
Maleimide
1.95
confidence
50
Bastadin 7
1.95
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.