BETABiohacksAI is a research tool for informational purposes only. All outputs are computational hypothesis candidates — not confirmed mechanisms, not medical advice, and not a substitute for professional medical judgment. Independent experimental validation is always required.
BiohacksAI is an evolving scientific literature platform. New compounds and evidence are indexed continuously.
B
MOLECULAR TARGETUniProt: P03372

ESR1

estrogen receptor 1

420 compounds · BiohacksAI corpus v20260307-01

420
compounds
Compounds
420
Gene Symbol
ESR1
NCBI Gene
2099

Looking for compounds that interact with ESR1?

View all 420 compounds →
About ESR1

ESR1 (estrogen receptor 1) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 420 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View ESR1 on UniProt →
Compounds Targeting ESR1 (50)
1
Tamoxifen
5.88
confidence
2
Raloxifene
4.77
confidence
3
Isoliquiritigenin
4.50
confidence
4
Coumaric Acid
4.42
confidence
5
Gossypol
4.42
confidence
6
Caffeic Acid Phenethyl Ester
4.25
confidence
7
Diethylstilbestrol
4.06
confidence
8
Emate
3.89
confidence
9
Phloretin
3.71
confidence
10
Afimoxifene
3.69
confidence
11
Trismethoxyresveratrol
3.56
confidence
292
studies
3.09
confidence
300
studies
3.09
confidence
298
studies
3.04
confidence
300
studies
3.00
confidence
300
studies
2.94
confidence
300
studies
2.94
confidence
18
Bithionol
2.89
confidence
19
Bazedoxifene
2.89
confidence
300
studies
2.83
confidence
21
Coumestrol
2.83
confidence
300
studies
2.77
confidence
300
studies
2.77
confidence
295
studies
2.77
confidence
25
Raloxifene Hydrochloride
2.77
confidence
300
studies
2.71
confidence
297
studies
2.71
confidence
298
studies
2.71
confidence
300
studies
2.71
confidence
30
Bisphenol A
2.71
confidence
31
Endoxifen
2.71
confidence
32
Tamoxifen Citrate
2.71
confidence
119
studies
2.64
confidence
34
Nandrolonepolycyclic
0
studies
2.64
confidence
300
studies
2.64
confidence
36
8z 345 Trimethoxystilbene
2.64
confidence
300
studies
2.56
confidence
300
studies
2.56
confidence
300
studies
2.56
confidence
300
studies
2.56
confidence
298
studies
2.56
confidence
297
studies
2.56
confidence
43
Diarylpropionitrile
2.56
confidence
44
Colchicineheterocyclic
0
studies
2.48
confidence
300
studies
2.48
confidence
300
studies
2.48
confidence
300
studies
2.48
confidence
298
studies
2.48
confidence
300
studies
2.48
confidence
50
Kurarinone
2.48
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.