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B
MOLECULAR TARGETUniProt: P25098

GRK2

G protein-coupled receptor kinase 2

125 compounds · BiohacksAI corpus v20260307-01

125
compounds
Compounds
125
Gene Symbol
GRK2
NCBI Gene
156

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About GRK2

GRK2 (G protein-coupled receptor kinase 2) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 125 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View GRK2 on UniProt →
Compounds Targeting GRK2 (50)
1
Paroxetine
4.39
confidence
2
Pf 03758309
3.00
confidence
3
Sangivamycin
3.00
confidence
4
Capivasertib
2.77
confidence
5
Balanol
2.30
confidence
6
Ravoxertinib
2.08
confidence
7
Gsk 180736a
2.08
confidence
8
Scutellaria Baicalensis
1.00
confidence
0
studies
1.00
confidence
10
Polygala Tenuifolia
1.00
confidence
11
Polygonum Cuspidatum
1.00
confidence
500
studies
1.00
confidence
13
Prunus Armeniaca
1.00
confidence
14
Prunus Persica
1.00
confidence
500
studies
1.00
confidence
16
Rehmannia Glutinosa
1.00
confidence
17
Salvia Miltiorrhiza
1.00
confidence
18
Scrophularia Ningpoensis
1.00
confidence
19
Agastache Rugosa
1.00
confidence
20
Allium Tuberosum
1.00
confidence
21
Aloe Vera
1.00
confidence
22
Apis Mellifera
1.00
confidence
23
Artemisia Capillaris
1.00
confidence
24
Aster Tataricus
1.00
confidence
25
Atractylodes Macrocephala
1.00
confidence
26
Bufo Bufo
1.00
confidence
27
Bupleurum Chinense
1.00
confidence
28
Carthamus Tinctorius
1.00
confidence
499
studies
1.00
confidence
30
Chaenomeles Speciosa
1.00
confidence
31
Citrus Reticulata
1.00
confidence
500
studies
1.00
confidence
33
Cuscuta Chinensis
1.00
confidence
34
Cynomorium Songaricum
1.00
confidence
35
Ephedra Sinica
1.00
confidence
36
Eriobotrya Japonica
1.00
confidence
37
Forsythia Suspensa
1.00
confidence
38
Gastrodia Elata
1.00
confidence
39
Glycine Max
1.00
confidence
40
Ligusticum Chuanxiong
1.00
confidence
41
Litchi Chinensis
1.00
confidence
42
Lithospermum Erythrorhizon
1.00
confidence
43
Lonicera Japonica
1.00
confidence
44
Morus Alba
1.00
confidence
0
studies
1.00
confidence
46
Paeonia Lactiflora
1.00
confidence
300
studies
1.00
confidence
48
Panax Notoginseng
1.00
confidence
49
Perilla Frutescens
1.00
confidence
50
Pinellia Ternata
1.00
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.