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B
MOLECULAR TARGETUniProt: P32298

GRK4

G protein-coupled receptor kinase 4

48 compounds · BiohacksAI corpus v20260307-01

48
compounds
Compounds
48
Gene Symbol
GRK4
NCBI Gene
2868

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About GRK4

GRK4 (G protein-coupled receptor kinase 4) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 48 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View GRK4 on UniProt →
Compounds Targeting GRK4 (48)
1
Erlotinib
5.55
confidence
2
Tozasertib
4.33
confidence
3
Ruxolitinib
4.23
confidence
4
Bosutinib
4.08
confidence
5
Midostaurin
3.85
confidence
6
Nintedanib
3.61
confidence
7
Tae 684
3.43
confidence
8
Fedratinib
3.40
confidence
9
Dovitinib
3.09
confidence
10
Lestaurtinib
3.04
confidence
11
Ruboxistaurin
2.94
confidence
12
R 406
2.83
confidence
13
Pha 665752
2.71
confidence
14
Kw 2449
2.64
confidence
15
Gsk 461364
2.40
confidence
16
Balanol
2.30
confidence
17
Su 014813
2.20
confidence
18
Tg100 115
2.08
confidence
298
studies
0.69
confidence
298
studies
0.69
confidence
500
studies
0.50
confidence
22
Aloe Vera
0.50
confidence
23
Apis Mellifera
0.50
confidence
24
Bombyx Mori
0.50
confidence
25
Bupleurum Chinense
0.50
confidence
26
Carthamus Tinctorius
0.50
confidence
27
Cimicifuga Heracleifolia
0.50
confidence
28
Citrus Reticulata
0.50
confidence
29
Coix Lacryma
0.50
confidence
30
Corydalis Yanhusuo
0.50
confidence
500
studies
0.50
confidence
32
Cuscuta Chinensis
0.50
confidence
33
Forsythia Suspensa
0.50
confidence
34
Hirudo Nipponia
0.50
confidence
35
Lindera Aggregata
0.50
confidence
36
Lonicera Japonica
0.50
confidence
300
studies
0.50
confidence
38
Perilla Frutescens
0.50
confidence
39
Pinellia Ternata
0.50
confidence
40
Polygonum Cuspidatum
0.50
confidence
500
studies
0.50
confidence
42
Prunella Vulgaris
0.50
confidence
43
Prunus Armeniaca
0.50
confidence
44
Prunus Mume
0.50
confidence
45
Scolopendra Subspinipes
0.50
confidence
46
Scutellaria Baicalensis
0.50
confidence
47
Smilax Glabra
0.50
confidence
48
Ziziphus Jujuba
0.50
confidence
Top 48 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.